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Items for "Radiolabeling"

Development of [103Pd]-labeled-bis(N4-methylthiosemicarbazone) complexes as possible therapeutic agents

Due to interesting tumor seeking properties of bis
-thiosemicarbazones, two radio palladium- bis -thiosemicarbazone complexes, i.e. , [ 103Pd]-pyruvaldehyde- bis(N4-methylthiosemicarbazone) ([ 103Pd] PTSM) and [ 103Pd]- di-acetyl-bis (N4-methylthiosemicarbazone) ([ 103Pd]ATSM) were prepared according to the analogy of radio copper homologs...

Keywords: Palladium-103, Palladium(II) complexes, Radiolabeling, bis-thiosemicarbazono complexes, PTSM

12/2006 | Radiochimica Acta, Oldenbourg Wissenschaftsverlag
Preparation, quality control and biodistribution studies of [67Ga]-DOTA-anti-CD20

Rituximab was successively labeled with [ 67Ga]-gallium chloride. The macrocyclic bifunctional chelating agent, N-succinimidyl-1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid (DOTA-NHS) was prepared at 25 °C using DOTA, N-hydroxy succinimide (NHS) in CH2Cl2...

Keywords: Rituximab, Gallium-67, Radiolabeling, Quality Control, DOTA

03/2008 | Radiochimica Acta, Oldenbourg Wissenschaftsverlag