Rituximab was successively labeled with [ 67Ga]-gallium chloride. The macrocyclic bifunctional chelating agent, N-succinimidyl-1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid (DOTA-NHS) was prepared at 25 °C using DOTA, N-hydroxy succinimide (NHS) in CH2Cl2...
Keywords: Rituximab, Gallium-67, Radiolabeling, Quality Control, DOTA
03/2008 | Radiochimica Acta, Oldenbourg Wissenschaftsverlag